PDB Information

PDB4J0S
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Optimization of 3,5-dimethylisoxazole derivatives as potent bromodomain ligands.
Hewings, D.S., Fedorov, O., Filippakopoulos, P., Martin, S., Picaud, S., Tumber, A., Wells, C., Olcina, M.M., Freeman, K., Gill, A., Ritchie, A.J., Sheppard, D.W., Russell, A.J., Hammond, E.M., Knapp, S., Brennan, P.E., Conway, S.J.
J.Med.Chem.
HeaderSignaling Protein
Released2013-01-31
Resolution1.840
CATH Insert Date28 Mar, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4j0sA01 10 Apr, 2013 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4