PDB Information

PDB4IWV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Optimising pharmacokinetics of glucokinase activators with matched triplicate design sets the discovery of AZD3651 and AZD9485
Waring, M.J., Bennett, S.N., Boyd, S., Campbell, L., Davies, R.D.M., Ogg, D.J., Hargreaves, D., Martin, N.G., Robb, G., Wilkinson, S., MacPaul, P., Wood, J.M.
To be Published
HeaderTransferase/Transferase Inhibitor
Released2013-01-24
Resolution2.100
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4iwvA01 09 Aug, 2013 3.40.367.20 Assigned
4iwvA02 09 Aug, 2013 3.30.420.40 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P35557 HXK4_HUMAN Homo sapiens Glucokinase