PDB Information

PDB4IUE
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Fragment-based ligand design of novel potent inhibitors of tankyrases.
Larsson, E.A., Jansson, A.E., Ng, F.M., Then, S.W., Panicker, R., Liu, B., Sangthongpitag, K., Pendharkar, V., Tai, S.J., Hill, J., Dan, C., Ho, S.Y., Cheong, W.W., Poulsen, A., Blanchard, S., Lin, G.R., Alam, J., Keller, T.H., Nordlund, P.
J.Med.Chem.
HeaderTransferase
Released2013-01-21
Resolution2.380
CATH Insert Date04 Aug, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Aug, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4iueA00 14 Aug, 2013 3.90.228.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2