PDB 4isu
PDB Information
| PDB | 4ISU |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Rattus norvegicus |
| Primary Citation | Studies on an (S)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor antagonist IKM-159: asymmetric synthesis, neuroactivity, and structural characterization.
J.Med.Chem.
|
| Header | Membrane Protein/Antagonist |
| Released | 2013-01-17 |
| Resolution | 2.300 |
| CATH Insert Date | 28 Mar, 2013 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 28 Mar, 2013 | Chopped |
| B | 28 Mar, 2013 | Chopped |
| C | 28 Mar, 2013 | Chopped |
| D | 28 Mar, 2013 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4isuA01 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuA02 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuB01 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuB02 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuC01 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuC02 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuD01 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
| 4isuD02 | 10 Apr, 2013 | 3.40.190.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P19491 | GRIA2_RAT | Rattus norvegicus | Glutamate receptor 2 |
| P19491 | GRIA2_RAT | Rattus norvegicus | Glutamate receptor 2 |
| P19491 | GRIA2_RAT | Rattus norvegicus | Glutamate receptor 2 |
| P19491 | GRIA2_RAT | Rattus norvegicus | Glutamate receptor 2 |
