PDB Information

PDB4IPF
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceXenopus laevis
Primary Citation
MDM2 Small-Molecule Antagonist RG7112 Activates p53 Signaling and Regresses Human Tumors in Preclinical Cancer Models.
Tovar, C., Graves, B., Packman, K., Filipovic, Z., Xia, B.H., Tardell, C., Garrido, R., Lee, E., Kolinsky, K., To, K.H., Linn, M., Podlaski, F., Wovkulich, P., Vu, B., Vassilev, L.T.
Cancer Res.
HeaderLigase/Antagonist
Released2013-01-09
Resolution1.700
CATH Insert Date28 Mar, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ipfA00 10 Apr, 2013 1.10.245.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P56273 MDM2_XENLA Xenopus laevis E3 ubiquitin-protein ligase Mdm2