PDB Information

PDB4IBM
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A highly selective dual insulin receptor (IR)/insulin-like growth factor 1 receptor (IGF-1R) inhibitor derived from an extracellular signal-regulated kinase (ERK) inhibitor.
Anastassiadis, T., Duong-Ly, K.C., Deacon, S.W., Lafontant, A., Ma, H., Devarajan, K., Dunbrack, R.L., Wu, J., Peterson, J.R.
J.Biol.Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-12-08
Resolution1.800
CATH Insert Date01 Sep, 2013

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped
B 02 Sep, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4ibmA01 10 Sep, 2013 3.30.200.20 Assigned
4ibmA02 10 Sep, 2013 1.10.510.10 Assigned
4ibmB01 10 Sep, 2013 3.30.200.20 Assigned
4ibmB02 10 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P06213 INSR_HUMAN Homo sapiens Insulin receptor
P06213 INSR_HUMAN Homo sapiens Insulin receptor