PDB Information

PDB4I41
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
A new target for an old drug: identifying mitoxantrone as a nanomolar inhibitor of PIM1 kinase via kinome-wide selectivity modeling.
Wan, X., Zhang, W., Li, L., Xie, Y., Li, W., Huang, N.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-11-27
Resolution2.700
CATH Insert Date15 Dec, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4i41A01 20 Dec, 2013 3.30.200.20 Assigned
4i41A02 20 Dec, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1