PDB 4hz0
PDB Information
PDB | 4HZ0 |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Escherichia coli |
Primary Citation | Pyrrolopyrimidine inhibitors of DNA gyrase B (GyrB) and topoisomerase IV (ParE). Part I: Structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity.
Bioorg.Med.Chem.Lett.
|
Header | Isomerase/Isomerase Inhibitor |
Released | 2012-11-14 |
Resolution | 2.200 |
CATH Insert Date | 28 Mar, 2013 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 Mar, 2013 | Chopped |
B | 28 Mar, 2013 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4hz0A00 | 01 Jul, 2013 | 3.30.565.10 | Assigned |
4hz0B00 | 01 Jul, 2013 | 3.30.565.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P20083 | PARE_ECOLI | Escherichia coli K-12 | DNA topoisomerase 4 subunit B |
P20083 | PARE_ECOLI | Escherichia coli K-12 | DNA topoisomerase 4 subunit B |