PDB Information

PDB4HY2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Development of cyclic peptomer inhibitors targeting the polo-box domain of polo-like kinase 1.
Murugan, R.N., Park, J.E., Lim, D., Ahn, M., Cheong, C., Kwon, T., Nam, K.Y., Choi, S.H., Kim, B.Y., Yoon, D.Y., Yaffe, M.B., Yu, D.Y., Lee, K.S., Bang, J.K.
Bioorg.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-11-12
Resolution2.000
CATH Insert Date07 Jul, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
D 08 Jul, 2013 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4hy2A01 09 Aug, 2013 3.30.1120.30 Assigned
4hy2A02 09 Aug, 2013 3.30.1120.30 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1