PDB 4hct
PDB Information
| PDB | 4HCT |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Covalent inhibitors of interleukin-2 inducible T cell kinase (itk) with nanomolar potency in a whole-blood assay.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2012-10-01 |
| Resolution | 1.480 |
| CATH Insert Date | 18 Nov, 2012 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 19 Nov, 2012 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4hctA01 | 02 Jan, 2013 | 3.30.200.20 | Assigned |
| 4hctA02 | 02 Jan, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |
