PDB Information

PDB4HAB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Development of cyclic peptomer inhibitors targeting the polo-box domain of polo-like kinase 1.
Murugan, R.N., Park, J.E., Lim, D., Ahn, M., Cheong, C., Kwon, T., Nam, K.Y., Choi, S.H., Kim, B.Y., Yoon, D.Y., Yaffe, M.B., Yu, D.Y., Lee, K.S., Bang, J.K.
Bioorg.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-09-26
Resolution2.650
CATH Insert Date07 Jul, 2013

PDB Images (13)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Chopped
D 08 Jul, 2013 Rejected
E 08 Jul, 2013 Rejected
F 08 Jul, 2013 Rejected

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4habA01 09 Aug, 2013 3.30.1120.30 Assigned
4habA02 09 Aug, 2013 3.30.1120.30 Assigned
4habB01 09 Aug, 2013 3.30.1120.30 Assigned
4habB02 09 Aug, 2013 3.30.1120.30 Assigned
4habC01 09 Aug, 2013 3.30.1120.30 Assigned
4habC02 09 Aug, 2013 3.30.1120.30 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1