PDB Information

PDB4H85
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Structure-based design and mechanisms of allosteric inhibitors for mitochondrial branched-chain alpha-ketoacid dehydrogenase kinase.
Tso, S.C., Qi, X., Gui, W.J., Chuang, J.L., Morlock, L.K., Wallace, A.L., Ahmed, K., Laxman, S., Campeau, P.M., Lee, B.H., Hutson, S.M., Tu, B.P., Williams, N.S., Tambar, U.K., Wynn, R.M., Chuang, D.T.
Proc.Natl.Acad.Sci.USA
HeaderTransferase/Transferase Inhibitor
Released2012-09-21
Resolution2.100
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4h85A01 09 Aug, 2013 1.20.140.20 Assigned
4h85A02 09 Aug, 2013 3.30.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q00972 BCKD_RAT Rattus norvegicus [3-methyl-2-oxobutanoate dehydrogenase [lipoamide]] kinase, mitochondrial