PDB Information

PDB4H6O
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceTrypanosoma cruzi
Primary Citation
Antitrypanosomal Lead Discovery: Identification of a Ligand-Efficient Inhibitor of Trypanosoma cruzi CYP51 and Parasite Growth.
Andriani, G., Amata, E., Beatty, J., Clements, Z., Coffey, B.J., Courtemanche, G., Devine, W., Erath, J., Juda, C.E., Wawrzak, Z., Wood, J.T., Lepesheva, G.I., Rodriguez, A., Pollastri, M.P.
J.Med.Chem.
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2012-09-19
Resolution2.800
CATH Insert Date28 Mar, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4h6oA00 10 Apr, 2013 1.10.630.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q7Z1V1 CP51_TRYCC Trypanosoma cruzi strain CL Brener Sterol 14-alpha demethylase