PDB Information

PDB4GS8
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, substrate-dependent modulators of insulin-degrading enzyme in amyloid-beta hydrolysis.
Charton, J., Gauriot, M., Guo, Q., Hennuyer, N., Marechal, X., Dumont, J., Hamdane, M., Pottiez, V., Landry, V., Sperandio, O., Flipo, M., Buee, L., Staels, B., Leroux, F., Tang, W.J., Deprez, B., Deprez-Poulain, R.
Eur.J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-08-27
Resolution2.990
CATH Insert Date15 Sep, 2013

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Sep, 2013 Chopped
B 16 Sep, 2013 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4gs8A01 30 Oct, 2013 3.30.830.10 Assigned
4gs8A02 30 Oct, 2013 3.30.830.10 Assigned
4gs8A03 30 Oct, 2013 3.30.830.10 Assigned
4gs8A04 30 Oct, 2013 3.30.830.10 Assigned
4gs8B01 30 Oct, 2013 3.30.830.10 Assigned
4gs8B02 30 Oct, 2013 3.30.830.10 Assigned
4gs8B03 30 Oct, 2013 3.30.830.10 Assigned
4gs8B04 30 Oct, 2013 3.30.830.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme