PDB Information

PDB4GRB
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo.
Dowling, J.E., Alimzhanov, M., Bao, L., Block, M.H., Chuaqui, C., Cooke, E.L., Denz, C.R., Hird, A., Huang, S., Larsen, N.A., Peng, B., Pontz, T.W., Rivard-Costa, C., Saeh, J.C., Thakur, K., Ye, Q., Zhang, T., Lyne, P.D.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2012-08-24
Resolution2.150
CATH Insert Date15 Sep, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Sep, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4grbA01 18 Sep, 2013 1.10.510.10 Assigned
4grbA02 18 Sep, 2013 3.30.200.20 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha