PDB 4gmb
PDB Information
| PDB | 4GMB |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of a Highly Potent, Cell-Permeable Macrocyclic Peptidomimetic (MM-589) Targeting the WD Repeat Domain 5 Protein (WDR5)-Mixed Lineage Leukemia (MLL) Protein-Protein Interaction.
J. Med. Chem.
|
| Header | Transcription/Transcription Inhibitor |
| Released | 2012-08-15 |
| Resolution | 2.780 |
| CATH Insert Date | 23 Feb, 2014 |
PDB Images (4)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 24 Feb, 2014 | Chopped |
| E | 24 Feb, 2014 | Rejected |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4gmbA00 | 07 Mar, 2014 | 2.130.10.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |
