PDB Information

PDB4GKM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis
Primary Citation
Repurposing the Chemical Scaffold of the Anti-Arthritic Drug Lobenzarit to Target Tryptophan Biosynthesis in Mycobacterium tuberculosis.
Evans, G.L., Gamage, S.A., Bulloch, E.M., Baker, E.N., Denny, W.A., Lott, J.S.
Chembiochem
HeaderTransferase/Transferase Inhibitor
Released2012-08-13
Resolution1.670
CATH Insert Date01 Sep, 2013

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped
B 02 Sep, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4gkmA01 04 Sep, 2013 1.20.970.10 Assigned
4gkmA02 04 Sep, 2013 3.40.1030.10 Assigned
4gkmB01 04 Sep, 2013 1.20.970.10 Assigned
4gkmB02 04 Sep, 2013 3.40.1030.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P9WFX5 TRPD_MYCTU Mycobacterium tuberculosis H37Rv Anthranilate phosphoribosyltransferase
P9WFX5 TRPD_MYCTU Mycobacterium tuberculosis H37Rv Anthranilate phosphoribosyltransferase