PDB Information

PDB4GK7
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Activity enhancement of the synthetic syrbactin proteasome inhibitor hybrid and biological evaluation in tumor cells.
Archer, C.R., Groll, M., Stein, M.L., Schellenberg, B., Clerc, J., Kaiser, M., Kondratyuk, T.P., Pezzuto, J.M., Dudler, R., Bachmann, A.S.
Biochemistry
HeaderHydrolase/Hydrolase Inhibitor
Released2012-08-10
Resolution2.800
CATH Insert Date04 Nov, 2012

PDB Images (63)

PDB Prints

PDB Chains (34)

Chain ID Date inserted into CATH CATH Status
1 05 Nov, 2012 Rejected
2 05 Nov, 2012 Rejected
3 05 Nov, 2012 Rejected
4 05 Nov, 2012 Rejected
5 05 Nov, 2012 Rejected
6 05 Nov, 2012 Rejected
a 05 Nov, 2012 Chopped
A 05 Nov, 2012 Chopped
b 05 Nov, 2012 Chopped
B 05 Nov, 2012 Chopped
C 05 Nov, 2012 Chopped
D 05 Nov, 2012 Chopped
E 05 Nov, 2012 Chopped
F 05 Nov, 2012 Chopped
G 05 Nov, 2012 Chopped
H 05 Nov, 2012 Chopped
I 05 Nov, 2012 Chopped
J 05 Nov, 2012 Chopped
K 05 Nov, 2012 Chopped
L 05 Nov, 2012 Chopped
M 05 Nov, 2012 Chopped
N 05 Nov, 2012 Chopped
O 05 Nov, 2012 Chopped
P 05 Nov, 2012 Chopped
Q 05 Nov, 2012 Chopped
R 05 Nov, 2012 Chopped
S 05 Nov, 2012 Chopped
T 05 Nov, 2012 Chopped
U 05 Nov, 2012 Chopped
V 05 Nov, 2012 Chopped
W 05 Nov, 2012 Chopped
X 05 Nov, 2012 Chopped
Y 05 Nov, 2012 Chopped
Z 05 Nov, 2012 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
4gk7a00 10 Nov, 2012 3.60.20.10 Assigned
4gk7A00 05 Feb, 2013 3.60.20.10 Assigned
4gk7b00 10 Nov, 2012 3.60.20.10 Assigned
4gk7B00 05 Feb, 2013 3.60.20.10 Assigned
4gk7C00 05 Feb, 2013 3.60.20.10 Assigned
4gk7D00 08 Feb, 2013 3.60.20.10 Assigned
4gk7E00 10 Nov, 2012 3.60.20.10 Assigned
4gk7F00 10 Nov, 2012 3.60.20.10 Assigned
4gk7G00 10 Nov, 2012 3.60.20.10 Assigned
4gk7H00 10 Nov, 2012 3.60.20.10 Assigned
4gk7I00 10 Nov, 2012 3.60.20.10 Assigned
4gk7J00 10 Nov, 2012 3.60.20.10 Assigned
4gk7K00 10 Nov, 2012 3.60.20.10 Assigned
4gk7L00 10 Nov, 2012 3.60.20.10 Assigned
4gk7M00 10 Nov, 2012 3.60.20.10 Assigned
4gk7N00 10 Nov, 2012 3.60.20.10 Assigned
4gk7O00 05 Feb, 2013 3.60.20.10 Assigned
4gk7P00 05 Feb, 2013 3.60.20.10 Assigned
4gk7Q00 05 Feb, 2013 3.60.20.10 Assigned
4gk7R00 08 Feb, 2013 3.60.20.10 Assigned
4gk7S00 10 Nov, 2012 3.60.20.10 Assigned
4gk7T00 10 Nov, 2012 3.60.20.10 Assigned
4gk7U00 10 Nov, 2012 3.60.20.10 Assigned
4gk7V00 10 Nov, 2012 3.60.20.10 Assigned
4gk7W00 10 Nov, 2012 3.60.20.10 Assigned
4gk7X00 10 Nov, 2012 3.60.20.10 Assigned
4gk7Y00 10 Nov, 2012 3.60.20.10 Assigned
4gk7Z00 10 Nov, 2012 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5