PDB Information

PDB4G9C
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Pyrazolopyridine inhibitors of B-Raf(V600E). Part 4: Rational design and kinase selectivity profile of cell potent type II inhibitors.
Wenglowsky, S., Moreno, D., Laird, E.R., Gloor, S.L., Ren, L., Risom, T., Rudolph, J., Sturgis, H.L., Voegtli, W.C.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2012-07-23
Resolution3.500
CATH Insert Date18 Nov, 2012

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 19 Nov, 2012 Chopped
B 19 Nov, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4g9cA01 02 Jan, 2013 3.30.200.20 Assigned
4g9cA02 02 Jan, 2013 1.10.510.10 Assigned
4g9cB01 02 Jan, 2013 3.30.200.20 Assigned
4g9cB02 02 Jan, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf
P15056 BRAF_HUMAN Homo sapiens Serine/threonine-protein kinase B-raf