PDB Information

PDB4G5P
MethodX-RAY DIFFRACTION
Host Organism
Gene SourceHomo sapiens
Primary Citation
Target Binding Properties and Cellular Activity of Afatinib (BIBW 2992), an Irreversible ErbB Family Blocker.
Solca, F., Dahl, G., Zoephel, A., Bader, G., Sanderson, M., Klein, C., Kraemer, O., Himmelsbach, F., Haaksma, E., Adolf, G.R.
J.Pharmacol.Exp.Ther.
HeaderTransferase/Transferase Inhibitor
Released2012-07-18
Resolution3.170
CATH Insert Date04 Nov, 2012

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped
B 05 Nov, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4g5pA01 25 Apr, 2013 3.30.200.20 Assigned
4g5pA02 25 Apr, 2013 1.10.510.10 Assigned
4g5pB01 25 Apr, 2013 3.30.200.20 Assigned
4g5pB02 25 Apr, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor
P00533 EGFR_HUMAN Homo sapiens Epidermal growth factor receptor