PDB 4fse
PDB Information
PDB | 4FSE |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Acyl guanidine inhibitors of beta-secretase (BACE-1): optimization of a micromolar hit to a nanomolar lead via iterative solid- and solution-phase library synthesis
J.Med.Chem.
|
Header | Hydrolase/Inhibitor |
Released | 2012-06-27 |
Resolution | 2.650 |
CATH Insert Date | 04 Nov, 2012 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 05 Nov, 2012 | Chopped |
B | 05 Nov, 2012 | Chopped |
D | 05 Nov, 2012 | Chopped |
E | 05 Nov, 2012 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4fseA01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseA02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseB01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseB02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseD01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseD02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseE01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4fseE02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |