PDB Information

PDB4EHR
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Pyrazole and pyrimidine phenylacylsulfonamides as dual Bcl-2/Bcl-xL antagonists.
Schroeder, G.M., Wei, D., Banfi, P., Cai, Z.W., Lippy, J., Menichincheri, M., Modugno, M., Naglich, J., Penhallow, B., Perez, H.L., Sack, J., Schmidt, R.J., Tebben, A., Yan, C., Zhang, L., Galvani, A., Lombardo, L.J., Borzilleri, R.M.
Bioorg.Med.Chem.Lett.
HeaderApoptosis
Released2012-04-03
Resolution2.090
CATH Insert Date10 Jun, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 10 Jun, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4ehrA00 26 Jul, 2013 Holding pen

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1