PDB Information

PDB4EFU
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Fragment-based discovery of hydroxy-indazole-carboxamides as novel small molecule inhibitors of Hsp90
Buchstaller, H.-P., Eggenweiler, H.-M., Sirrenberg, C., Graedler, U., Musil, D., Hoppe, E., Zimmermann, A., Schwartz, H., Maerz, J., Bomke, J., Wegener, A., Wolf, M.
Bioorg.Med.Chem.Lett.
HeaderChaperone/Chaperone Inhibitor
Released2012-03-30
Resolution2.000
CATH Insert Date04 Nov, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4efuA00 31 Aug, 2013 3.30.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P07900 HS90A_HUMAN Homo sapiens Heat shock protein HSP 90-alpha