PDB Information

PDB4E73
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Identification of an Adamantyl Azaquinolone JNK Selective Inhibitor.
Haynes, N.E., Scott, N.R., Chen, L.C., Janson, C.A., Li, J.K., Lukacs, C.M., Railkar, A., Tozzo, E., Whittard, T., Brown, N.F., Cheung, A.W.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2012-03-16
Resolution2.270
CATH Insert Date07 Jul, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4e73A01 09 Aug, 2013 3.30.200.20 Assigned
4e73A02 09 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9UQF2 JIP1_HUMAN Homo sapiens C-Jun-amino-terminal kinase-interacting protein 1
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8