PDB Information

PDB4E67
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Using ligand-mapping simulations to design a ligand selectively targeting a cryptic surface pocket of polo-like kinase 1.
Tan, Y.S., Sledz, P., Lang, S., Stubbs, C.J., Spring, D.R., Abell, C., Best, R.B.
Angew.Chem.Int.Ed.Engl.
HeaderTransferase/Transferase Inhibitor
Released2012-03-15
Resolution2.100
CATH Insert Date04 Nov, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped
B 05 Nov, 2012 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4e67A01 10 Nov, 2012 3.30.1120.30 Assigned
4e67A02 10 Nov, 2012 3.30.1120.30 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53350 PLK1_HUMAN Homo sapiens Serine/threonine-protein kinase PLK1