PDB 4dw6
PDB Information
| PDB | 4DW6 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Mycobacterium tuberculosis |
| Primary Citation | Discovery of novel N-phenylphenoxyacetamide derivatives as EthR inhibitors and ethionamide boosters by combining high-throughput screening and synthesis.
J.Med.Chem.
|
| Header | Transcription/Inhibitor |
| Released | 2012-02-24 |
| Resolution | 2.000 |
| CATH Insert Date | 07 Jul, 2013 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Jul, 2013 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4dw6A01 | 08 Aug, 2013 | 1.10.10.60 | Assigned |
| 4dw6A02 | 08 Aug, 2013 | 1.10.357.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P9WMC1 | ETHR_MYCTU | Mycobacterium tuberculosis H37Rv | HTH-type transcriptional regulator EthR |
