PDB Information

PDB4DTT
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, substrate-dependent modulators of insulin-degrading enzyme in amyloid-beta hydrolysis.
Charton, J., Gauriot, M., Guo, Q., Hennuyer, N., Marechal, X., Dumont, J., Hamdane, M., Pottiez, V., Landry, V., Sperandio, O., Flipo, M., Buee, L., Staels, B., Leroux, F., Tang, W.J., Deprez, B., Deprez-Poulain, R.
Eur.J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-02-21
Resolution3.220
CATH Insert Date28 Mar, 2013

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped
B 28 Mar, 2013 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
4dttA01 31 Aug, 2013 3.30.830.10 Assigned
4dttA02 31 Aug, 2013 3.30.830.10 Assigned
4dttA03 31 Aug, 2013 3.30.830.10 Assigned
4dttA04 31 Aug, 2013 3.30.830.10 Assigned
4dttB01 31 Aug, 2013 3.30.830.10 Assigned
4dttB02 31 Aug, 2013 3.30.830.10 Assigned
4dttB03 31 Aug, 2013 3.30.830.10 Assigned
4dttB04 31 Aug, 2013 3.30.830.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme
P14735 IDE_HUMAN Homo sapiens Insulin-degrading enzyme