PDB Information

PDB4DIJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The central valine concept provides an entry in a new class of non peptide inhibitors of the p53-MDM2 interaction.
Furet, P., Chene, P., De Pover, A., Valat, T.S., Lisztwan, J.H., Kallen, J., Masuya, K.
Bioorg.Med.Chem.Lett.
HeaderLigase/Ligase Inhibitor
Released2012-01-31
Resolution1.900
CATH Insert Date27 May, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 May, 2012 Chopped
B 28 May, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4dijA00 08 Jun, 2012 1.10.245.10 Assigned
4dijB00 08 Jun, 2012 1.10.245.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q00987 MDM2_HUMAN Homo sapiens E3 ubiquitin-protein ligase Mdm2
Q00987 MDM2_HUMAN Homo sapiens E3 ubiquitin-protein ligase Mdm2