PDB Information

PDB4D0X
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Pyrrole-3-Carboxamides as Potent and Selective Jak2 Inhibitors.
Brasca, M.G., Nesi, M., Avanzi, N., Ballinari, D., Bandiera, T., Bertrand, J., Bindi, S., Canevari, G., Carenzi, D., Casero, D., Ceriani, L., Ciomei, M., Cirla, A., Colombo, M., Cribioli, S., Cristiani, C., Della Vedova, F., Fachin, G., Fasolini, M., Felder, E.R., Galvani, A., Isacchi, A., Mirizzi, D., Motto, I., Panzeri, A., Pesenti, E., Vianello, P., Gnocchi, P., Donati, D.
Bioorg.Med.Chem.
HeaderTransferase
Released2014-04-30
Resolution1.820
CATH Insert Date10 Aug, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Aug, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4d0xA01 19 Aug, 2014 3.30.200.20 Assigned
4d0xA02 19 Aug, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2