PDB 4d09
PDB Information
PDB | 4D09 |
Method | X-RAY DIFFRACTION |
Host Organism | SPODOPTERA FRUGIPERDA |
Gene Source | HOMO SAPIENS |
Primary Citation | Structure-Based Design of a Potent, Selective, and Brain Penetrating Pde2 Inhibitor with Demonstrated Target Engagement.
Acs Med.Chem.Lett.
|
Header | Hydrolase |
Released | 2014-04-24 |
Resolution | 2.500 |
CATH Insert Date | 24 Aug, 2014 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 25 Aug, 2014 | Chopped |
B | 25 Aug, 2014 | Chopped |
C | 25 Aug, 2014 | Chopped |
D | 25 Aug, 2014 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4d09A00 | 27 Aug, 2014 | 1.10.1300.10 | Assigned |
4d09B00 | 27 Aug, 2014 | 1.10.1300.10 | Assigned |
4d09C00 | 27 Aug, 2014 | 1.10.1300.10 | Assigned |
4d09D00 | 27 Aug, 2014 | 1.10.1300.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O00408 | PDE2A_HUMAN | Homo sapiens | cGMP-dependent 3',5'-cyclic phosphodiesterase |
O00408 | PDE2A_HUMAN | Homo sapiens | cGMP-dependent 3',5'-cyclic phosphodiesterase |
O00408 | PDE2A_HUMAN | Homo sapiens | cGMP-dependent 3',5'-cyclic phosphodiesterase |
O00408 | PDE2A_HUMAN | Homo sapiens | cGMP-dependent 3',5'-cyclic phosphodiesterase |