PDB Information

PDB4CSJ
MethodX-RAY DIFFRACTION
Host OrganismTRICHOPLUSIA NI
Gene SourceHOMO SAPIENS
Primary Citation
The Discovery of Potent and Selective Non-Steroidal Glucocorticoid Receptor Modulators, Suitable for Inhalation.
Edman, K., Ahlgren, R., Bengtsson, M., Bladh, H., Backstrom, S., Dahmen, J., Henriksson, K., Hillertz, P., Hulikal, V., Jerre, A., Kinchin, L., Kase, C., Lepisto, M., Mile, I., Nilsson, S., Smailagic, A., Taylor, J., Tjornebo, A., Wissler, L., Hansson, T.
Bioorg.Med.Chem.Lett.
HeaderSignaling Protein
Released2014-03-07
Resolution2.300
CATH Insert Date11 May, 2014

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 12 May, 2014 Chopped
B 12 May, 2014 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4csjA00 17 May, 2014 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04150 GCR_HUMAN Homo sapiens Glucocorticoid receptor
Q15596 NCOA2_HUMAN Homo sapiens Nuclear receptor coactivator 2