PDB Information

PDB4CBY
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Design, synthesis, and biological evaluation of potent and selective class IIa histone deacetylase (HDAC) inhibitors as a potential therapy for Huntington's disease.
Burli, R.W., Luckhurst, C.A., Aziz, O., Matthews, K.L., Yates, D., Lyons, K.A., Beconi, M., McAllister, G., Breccia, P., Stott, A.J., Penrose, S.D., Wall, M., Lamers, M., Leonard, P., Muller, I., Richardson, C.M., Jarvis, R., Stones, L., Hughes, S., Wishart, G., Haughan, A.F., O'Connell, C., Mead, T., McNeil, H., Vann, J., Mangette, J., Maillard, M., Beaumont, V., Munoz-Sanjuan, I., Dominguez, C.
J. Med. Chem.
HeaderHydrolase
Released2013-10-17
Resolution2.720
CATH Insert Date15 Dec, 2013

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2013 Chopped
B 16 Dec, 2013 Chopped
C 16 Dec, 2013 Chopped
D 16 Dec, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4cbyA00 20 Dec, 2013 3.40.800.20 Assigned
4cbyB00 20 Dec, 2013 3.40.800.20 Assigned
4cbyC00 20 Dec, 2013 3.40.800.20 Assigned
4cbyD00 20 Dec, 2013 3.40.800.20 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4
P56524 HDAC4_HUMAN Homo sapiens Histone deacetylase 4