PDB Information

PDB4BUS
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Para-Substituted 2-Phenyl-3,4-Dihydroquinazolin-4-Ones as Potent and Selective Tankyrase Inhibitors.
Haikarainen, T., Koivunen, J., Narwal, M., Venkannagari, H., Obaji, E., Joensuu, P., Pihlajaniemi, T., Lehtio, L.
Chemmedchem
HeaderTransferase
Released2013-06-24
Resolution1.900
CATH Insert Date03 Nov, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 04 Nov, 2013 Chopped
B 04 Nov, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4busA00 08 Nov, 2013 3.90.228.10 Assigned
4busB00 08 Nov, 2013 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2