PDB Information

PDB4BJK
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceTRYPANOSOMA BRUCEI
Primary Citation
Rational Development of 4-Aminopyridyl-Based Inhibitors Targeting Trypanosoma Cruzi Cyp51 as Anti-Chagas Agents.
Choi, J.Y., Calvet, C.M., Gunatilleke, S.S., Ruiz, C., Cameron, M.D., Mckerrow, J.H., Podust, L.M., Roush, W.R.
J.Med.Chem.
HeaderOxidoreductase
Released2013-04-18
Resolution2.670
CATH Insert Date22 Sep, 2013

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 23 Sep, 2013 Chopped
B 23 Sep, 2013 Chopped
C 23 Sep, 2013 Chopped
D 23 Sep, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4bjkA00 25 Sep, 2013 1.10.630.10 Assigned
4bjkB00 25 Sep, 2013 1.10.630.10 Assigned
4bjkC00 25 Sep, 2013 1.10.630.10 Assigned
4bjkD00 25 Sep, 2013 1.10.630.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q385E8 Q385E8_TRYB2 Trypanosoma brucei brucei TREU927 Lanosterol 14-alpha-demethylase
Q385E8 Q385E8_TRYB2 Trypanosoma brucei brucei TREU927 Lanosterol 14-alpha-demethylase
Q385E8 Q385E8_TRYB2 Trypanosoma brucei brucei TREU927 Lanosterol 14-alpha-demethylase
Q385E8 Q385E8_TRYB2 Trypanosoma brucei brucei TREU927 Lanosterol 14-alpha-demethylase