PDB 4bcq
PDB Information
| PDB | 4BCQ |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Comparative Structural and Functional Studies of 4-(Thiazol- 5-Yl)-2-(Phenylamino)Pyrimidine-5-Carbonitrile Cdk9 Inhibitors Suggest the Basis for Isotype Selectivity.
J.Med.Chem.
|
| Header | Transferase/Cell Cycle |
| Released | 2012-10-02 |
| Resolution | 2.400 |
| CATH Insert Date | 20 Jan, 2013 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 21 Jan, 2013 | Chopped |
| B | 21 Jan, 2013 | Chopped |
| C | 21 Jan, 2013 | Chopped |
| D | 21 Jan, 2013 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4bcqA01 | 11 Feb, 2013 | 3.30.200.20 | Assigned |
| 4bcqA02 | 11 Feb, 2013 | 1.10.510.10 | Assigned |
| 4bcqB01 | 24 Jan, 2013 | 1.10.472.10 | Assigned |
| 4bcqB02 | 24 Jan, 2013 | 1.10.472.10 | Assigned |
| 4bcqC01 | 11 Feb, 2013 | 3.30.200.20 | Assigned |
| 4bcqC02 | 11 Feb, 2013 | 1.10.510.10 | Assigned |
| 4bcqD01 | 24 Jan, 2013 | 1.10.472.10 | Assigned |
| 4bcqD02 | 24 Jan, 2013 | 1.10.472.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
| P30274 | CCNA2_BOVIN | Bos taurus | Cyclin-A2 |
| P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
| P30274 | CCNA2_BOVIN | Bos taurus | Cyclin-A2 |
