PDB 4bcg
PDB Information
| PDB | 4BCG |
| Method | X-RAY DIFFRACTION |
| Host Organism | SPODOPTERA FRUGIPERDA |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Substituted 4-(Thiazol-5-Yl)-2-(Phenylamino)Pyrimidines are Highly Active Cdk9 Inhibitors: Synthesis, X-Ray Crystal Structure, Sar and Anti-Cancer Activities.
J.Med.Chem.
|
| Header | Transferase/Cell Cycle |
| Released | 2012-10-02 |
| Resolution | 3.090 |
| CATH Insert Date | 07 Jul, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Jul, 2013 | Chopped |
| B | 08 Jul, 2013 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4bcgA01 | 09 Aug, 2013 | 3.30.200.20 | Assigned |
| 4bcgA02 | 09 Aug, 2013 | 1.10.510.10 | Assigned |
| 4bcgB01 | 09 Aug, 2013 | 1.10.472.10 | Assigned |
| 4bcgB02 | 09 Aug, 2013 | 1.10.472.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60563 | CCNT1_HUMAN | Homo sapiens | Cyclin-T1 |
| P50750 | CDK9_HUMAN | Homo sapiens | Cyclin-dependent kinase 9 |
