PDB Information

PDB4AZF
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Selectivity, Co-Crystal Structures and Neuroprotective Properties of Leucettines, a Family of Protein Kinase Inhibitors Derived from the Marine Sponge Alkaloid Leucettamine B.
Tahtouh, T., Elkins, J.M., Filippakopoulos, P., Soundararajan, M., Burgy, G., Durieu, E., Cochet, C., Schmid, R.S., Lo, D.C., Delhommel, F., Oberholzer, A., Laurence, P., Carreaux, F., Bazureau, J.P., Knapp, S., Meijer, L.
J.Med.Chem.
HeaderTransferase
Released2012-06-25
Resolution2.550
CATH Insert Date04 Nov, 2012

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4azfA01 23 Jul, 2013 3.30.10.30 Assigned
4azfA02 23 Jul, 2013 3.30.200.20 Assigned
4azfA03 23 Jul, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q92630 DYRK2_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 2