PDB 4a9o
PDB Information
| PDB | 4A9O |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Fragment-Based Discovery of Bromodomain Inhibitors Part 2: Optimization of Phenylisoxazole Sulfonamides.
J.Med.Chem.
|
| Header | Signaling Protein/Inhibitor |
| Released | 2011-11-26 |
| Resolution | 1.780 |
| CATH Insert Date | 12 Feb, 2012 |
PDB Images (7)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 13 Feb, 2012 | Chopped |
| B | 13 Feb, 2012 | Chopped |
| C | 13 Feb, 2012 | Chopped |
CATH Domains (3)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4a9oA00 | 16 Feb, 2012 | 1.20.920.10 | Assigned |
| 4a9oB00 | 15 Feb, 2012 | 1.20.920.10 | Assigned |
| 4a9oC00 | 16 Feb, 2012 | 1.20.920.10 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P25440 | BRD2_HUMAN | Homo sapiens | Bromodomain-containing protein 2 |
| P25440 | BRD2_HUMAN | Homo sapiens | Bromodomain-containing protein 2 |
| P25440 | BRD2_HUMAN | Homo sapiens | Bromodomain-containing protein 2 |
