PDB Information

PDB4A9H
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Fragment-Based Discovery of Bromodomain Inhibitors Part 1: Inhibitor Binding Modes and Implications for Lead Discovery.
Chung, C.W., Dean, T.W., Woolven, J.M., Bamborough, P.
J.Med.Chem.
HeaderSignaling Protein
Released2011-11-26
Resolution2.050
CATH Insert Date15 Jan, 2012

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 16 Jan, 2012 Chopped
B 16 Jan, 2012 Chopped
C 16 Jan, 2012 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4a9hA00 19 Jan, 2012 1.20.920.10 Assigned
4a9hB00 19 Jan, 2012 1.20.920.10 Assigned
4a9hC00 19 Jan, 2012 1.20.920.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2