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PDB Information
| PDB | 4A9E |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | HOMO SAPIENS |
| Primary Citation |
Fragment-Based Discovery of Bromodomain Inhibitors Part 1: Inhibitor Binding Modes and Implications for Lead Discovery.
Chung, C.W., Dean, A.W., Woolven, J.M., Bamborough, P.
J.Med.Chem.
|
| Header | Signaling Protein |
| Released | 2011-11-26 |
| Resolution | 1.910 |
| CATH Insert Date | 15 Jan, 2012 |
PDB Images (7)
4a9eA00
CATH Domain 4a9eA00
4a9eB00
CATH Domain 4a9eB00
4a9eC00
CATH Domain 4a9eC00
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
| A | 16 Jan, 2012 | Chopped
|
| B | 16 Jan, 2012 | Chopped
|
| C | 16 Jan, 2012 | Chopped
|
CATH Domains (3)
UniProtKB Entries (3)
| Accession |
Gene ID |
Taxon |
Description |
| P25440 |
BRD2_HUMAN |
Homo sapiens |
Bromodomain-containing protein 2 |
| P25440 |
BRD2_HUMAN |
Homo sapiens |
Bromodomain-containing protein 2 |
| P25440 |
BRD2_HUMAN |
Homo sapiens |
Bromodomain-containing protein 2 |