PDB Information

PDB4A7C
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Hit to Lead Evaluation of 1,2,3-Triazolo[4,5-B]Pyridines as Pim Kinase Inhibitors.
Pastor, J., Oyarzabal, J., Saluste, G., Alvarez, R.M., Rivero, V., Ramos, F., Cendon, E., Blanco-Aparicio, C., Ajenjo, N., Cebria, A., Albarran, M.I., Cebrian, D., Corrionero, A., Fominaya, J., Montoya, G., Mazzorana, M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2011-11-12
Resolution2.300
CATH Insert Date19 Feb, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Feb, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4a7cA01 22 Feb, 2012 3.30.200.20 Assigned
4a7cA02 22 Feb, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1