PDB Information

PDB3ZMM
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of Novel Jak2-Stat Pathway Inhibitors with Extended Residence Time on Target.
Guan, H., Lamb, M.L., Peng, B., Huang, S., Degrace, N., Read, J., Hussain, S., Wu, J., Rivard, C., Alimzhanov, M., Bebernitz, G., Bell, K., Ye, M., Zinda, M., Ioannidis, S.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2013-02-11
Resolution2.510
CATH Insert Date07 Jul, 2013

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3zmmA01 09 Aug, 2013 3.30.200.20 Assigned
3zmmA02 09 Aug, 2013 1.10.510.10 Assigned
3zmmB01 09 Aug, 2013 3.30.200.20 Assigned
3zmmB02 09 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2
O60674 JAK2_HUMAN Homo sapiens Tyrosine-protein kinase JAK2