PDB 3wzk
PDB Information
| PDB | 3WZK |
| Method | X-RAY DIFFRACTION |
| Host Organism | CELL-FREE SYNTHESIS |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of Imidazo[1,2-b]pyridazine Derivatives: Selective and Orally Available Mps1 (TTK) Kinase Inhibitors Exhibiting Remarkable Antiproliferative Activity
J.Med.Chem.
|
| Header | Transferase |
| Released | 2014-09-29 |
| Resolution | 2.300 |
| CATH Insert Date | 28 Jun, 2015 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Jun, 2015 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3wzkA01 | 10 Jul, 2015 | 3.30.200.20 | Assigned |
| 3wzkA02 | 10 Jul, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P33981 | TTK_HUMAN | Homo sapiens | Dual specificity protein kinase TTK |
