PDB 3ws8
PDB Information
| PDB | 3WS8 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stability.
Bioorg.Med.Chem.
|
| Header | Hydrolase/Hydrolase Inhibitor |
| Released | 2014-03-04 |
| Resolution | 2.600 |
| CATH Insert Date | 15 Jun, 2014 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Jun, 2014 | Chopped |
| B | 16 Jun, 2014 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3ws8A00 | 18 Jun, 2014 | 1.10.1300.10 | Assigned |
| 3ws8B00 | 18 Jun, 2014 | 1.10.1300.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q9Y233 | PDE10_HUMAN | Homo sapiens | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
| Q9Y233 | PDE10_HUMAN | Homo sapiens | cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A |
