PDB Information

PDB3WIZ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of potent Mcl-1/Bcl-xL dual inhibitors by using a hybridization strategy based on structural analysis of target proteins.
Tanaka, Y., Aikawa, K., Nishida, G., Homma, M., Sogabe, S., Igaki, S., Hayano, Y., Sameshima, T., Miyahisa, I., Kawamoto, T., Tawada, M., Imai, Y., Inazuka, M., Cho, N., Imaeda, Y., Ishikawa, T.
J.Med.Chem.
HeaderApoptosis
Released2013-09-26
Resolution2.450
CATH Insert Date01 Dec, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 02 Dec, 2013 Chopped
B 02 Dec, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3wizA00 04 Dec, 2013 Holding pen
3wizB00 04 Dec, 2013 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1