PDB Information

PDB3UR4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5.
Senisterra, G., Wu, H., Allali-Hassani, A., Wasney, G.A., Barsyte-Lovejoy, D., Dombrovski, L., Dong, A., Nguyen, K.T., Smil, D., Bolshan, Y., Hajian, T., He, H., Seitova, A., Chau, I., Li, F., Poda, G., Couture, J.F., Brown, P.J., Al-Awar, R., Schapira, M., Arrowsmith, C.H., Vedadi, M.
Biochem. J.
HeaderTranscription/Inhibitor
Released2011-11-21
Resolution1.800
CATH Insert Date08 Jan, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2012 Chopped
B 09 Jan, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3ur4A00 17 Jul, 2013 2.130.10.10 Assigned
3ur4B00 17 Jul, 2013 2.130.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P61964 WDR5_HUMAN Homo sapiens WD repeat-containing protein 5
P61964 WDR5_HUMAN Homo sapiens WD repeat-containing protein 5