PDB Information

PDB3ULI
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of azabenzimidazole derivatives as potent, selective inhibitors of TBK1/IKK epsilon kinases.
Wang, T., Block, M.A., Cowen, S., Davies, A.M., Devereaux, E., Gingipalli, L., Johannes, J., Larsen, N.A., Su, Q., Tucker, J.A., Whitston, D., Wu, J., Zhang, H.J., Zinda, M., Chuaqui, C.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-11-10
Resolution2.000
CATH Insert Date01 Sep, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3uliA01 03 Sep, 2013 3.30.200.20 Assigned
3uliA02 03 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2