PDB Information

PDB3UH2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure of human tankyrase 1 in complex with small-molecule inhibitors PJ34 and XAV939.
Kirby, C.A., Cheung, A., Fazal, A., Shultz, M.D., Stams, T.
Acta Crystallogr.,Sect.F
HeaderTransferase/Transferase Inhibitor
Released2011-11-03
Resolution2.000
CATH Insert Date19 Feb, 2012

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 20 Feb, 2012 Chopped
B 20 Feb, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3uh2A00 22 Feb, 2012 3.90.228.10 Assigned
3uh2B00 23 Feb, 2012 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1
O95271 TNKS1_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-1