PDB Information

PDB3UA8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
6-Amino quinazolinedione sulfonamides as orally active competitive AMPA receptor antagonists.
Orain, D., Ofner, S., Koller, M., Carcache, D.A., Froestl, W., Allgeier, H., Rasetti, V., Nozulak, J., Mattes, H., Soldermann, N., Floersheim, P., Desrayaud, S., Kallen, J., Lingenhoehl, K., Urwyler, S.
Bioorg.Med.Chem.Lett.
HeaderTransport Protein/Antagonist
Released2011-10-21
Resolution1.900
CATH Insert Date15 Jan, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Jan, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3ua8A01 19 Jan, 2012 3.40.190.10 Assigned
3ua8A02 19 Jan, 2012 3.40.190.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P42262 GRIA2_HUMAN Homo sapiens Glutamate receptor 2