PDB Information

PDB3U5K
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
Filippakopoulos, P., Picaud, S., Fedorov, O., Keller, M., Wrobel, M., Morgenstern, O., Bracher, F., Knapp, S.
Bioorg.Med.Chem.
HeaderSignaling Protein/Inhibitor
Released2011-10-11
Resolution1.800
CATH Insert Date27 Nov, 2011

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped
B 29 Nov, 2011 Chopped
C 29 Nov, 2011 Chopped
D 29 Nov, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3u5kA01 01 Dec, 2011 1.20.920.10 Assigned
3u5kB01 01 Dec, 2011 1.20.920.10 Assigned
3u5kC01 01 Dec, 2011 1.20.920.10 Assigned
3u5kD01 01 Dec, 2011 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4